PCAF-IN-2 (compound 17) is a potent PCAF inhibitor with an IC 50 value of 5.31 µM. PCAF-IN-2 shows anti-tumour activity. CAF-IN-2 induces apoptosis and arrest the cell cycle at the G2/M phaseIn VitroPCAF-IN-2 shows anti-tumour activity with IC 50 s of 3.06, 5.69, 7.56, 2.83 µM for HePG2, MCF-7, PC3, HCT-116 cells, respectively. PCAF-IN-2 (10 µM; 24 h) induces apoptosis and arrest the cell cycle at the G2/M phase in HePG2 cells. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:PCAF 5.31 μM (IC 50 ).
Specifications and Purity: ≥98%
Molecular Formula: C10H7F3N6
Molecular Weight: 268.20
- UPC:
- 42222103
- Condition:
- New
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- P650341-25mg
- CAS:
- 56173-05-8
- Product Size:
- 25mg
akash.verma@cenmed.com
(732) 447-1115





