N-Desmethyl Pirenzepine-d8 is a deuterium-labeled metabolite of Pirenzepine (sc-204197). Pirenzepine is a selective antagonist for the M1 muscarinic receptor (mAChR) and is reported to block presynaptic M1 receptors as well as some reported inverse agonist activity. A study investigating the pharmacological characterization of the muscarinic receptors associated with ACh-induced pulmonary vasodilation in a rabbit model of pulmonary hypertension determined the IC|50|to be 2.51x10|-7|M. Additional research studies have investigated the role of Pirenzepine in the pathophysiology of myopia. Other M1 receptor antagonists offered include Telenzepine (sc-204332).N-Desmethyl Pirenzepine-d8is a deuterium-labeled metabolite of Pirenzepine.
Molecular Formula: C18H11D8N5O2
Molecular Weight: 345.43
PubChem CID: 46781185
- UPC:
- 51151504
- Condition:
- New
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- N379375-1mg
- CAS:
- 1189860-05-6
- Product Size:
- 1mg
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