Enzalutamide carboxylic acid (MDV3100 carboxylic acid) is an inactive metabolite of Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist.In VitroEnzalutamide is converted into its major metabolites, N-desmethyl enzalutamide and carboxylic acid enzalutamide, by cytochrome P450 (CYP) 3A4/5 and CYP2C8, respectively. N-desmethyl enzalutamide has clinically relevant anti-androgen capacities similar to enzalutamide, whereas carboxylic acid enzalutamide is inactive. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:Solid.
Specifications and Purity: ≥98%
Molecular Formula: C20H13F4N3O3S
Molecular Weight: 451.39
PubChem CID: 46898522
Isomeric SMILES: CC1(C(=O)N(C(=S)N1C2=CC(=C(C=C2)C(=O)O)F)C3=CC(=C(C=C3)C#N)C(F)(F)F)C
- UPC:
- 51241105
- Condition:
- New
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- E650376-5mg
- CAS:
- 1242137-15-0
- Product Size:
- 5mg
akash.verma@cenmed.com
(732) 447-1115





