EGFR-IN-69 (compound 17g) is a potent EGFR inhibitor, with IC 50 values of 4.3, 6.6 and 25.6 nM against EGFR L858R/T790M/C797S , EGFR L858R/T790M , and EGFR 19del/T790M/C797S , respectively. EGFR-IN-69 can be used for non-small-cell-lung-cancer (NSCLC) researchForm:SolidIC50& Target:EGFR L858R/T790M/C797S 4.3 ± 0.9 nM (IC 50 ) EGFR L858R/T790M 6.6 ± 0.8 nM (IC 50 ) EGFR del19 T790M C797S 25.6 ± 7.5 nM (IC 50 ) EGFR WT 816.0 ± 82 nM (IC 50 ).
Specifications and Purity: ≥99%
Molecular Formula: C31H37Cl2N7O3S
Molecular Weight: 658.64
- UPC:
- 51131508
- Condition:
- New
- HazmatClass:
- No
- WeightUOM:
- LB
- MPN:
- E647157-25mg
- CAS:
- 2433837-65-9
- Product Size:
- 25mg
akash.verma@cenmed.com
(732) 447-1115





