A non-cholestatic regioisomer of E217G that acts as a substrate for MRP2, competing with E217G for MRP2-mediated transport (IC<sub>50</sub> = 14.2 µM).
A non-cholestatic regioisomer of E217G that acts as a substrate for MRP2, competing with E217G for MRP2-mediated transport (IC<sub>50</sub> = 14.2 µM).
A metabolite of estradiol 3-sulfate that has been modified by a UDP-glucuronosyltransferase enhances utilization by anion transporters, most commonly leading to excretion in urine and bile.
A metabolite of estradiol 3-sulfate that has been modified by a UDP-glucuronosyltransferase enhances utilization by anion transporters, most commonly leading to excretion in urine and bile.