D,L-Venlafaxine (C007B-137870)

D,L-Venlafaxine is an isomer of Venlafaxine . Venlafaxine is a derivative of phenylethylamine which is reported to facilitate neurotransmission within the central nervous system via blocking the presynaptic reuptake of neuroamines such as serotonin (5-hydroxytryptamine; 5-HT) and noradrenaline (norepinephrine). Velanfaxine is also reported to be a weak inhibitor of dopamine reuptake.|In vitro|studies indicate that Venlafaxine does not demonstrate significant activity for muscarinic, histaminergic or α-1 adrenergic receptors. The metabolism of venlafaxine is reported to occur by cytochrome P450 (CYP) enzyme CYP2D6 yielding O-desmethylvenlafaxine. A lesser metabolite, N-desmethylvenlafaxine is produced by CYP3A4.

Specifications and Purity: 10mM in DMSO

Molecular Formula: C17H27NO2

Molecular Weight: 277.4

PubChem CID: 5656

Isomeric SMILES: CN(C)CC(C1=CC=C(C=C1)OC)C2(CCCCC2)O

Beilstein Registry Number: 4234848