TX1-85-1 (C007B-430252)

Catalog No.: C007B-430252
Manufacturer No.: T646130-1mg
Manufacturer Name: Aladdin Scientific
Quantity: 1
Unit of Measure: EA

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Description
Specifications

TX1-85-1 is an irreversible Her3 (ErbB3) inhibitor with an IC 50 of 23 nM. TX1-85-1 is also the first selective Her3 ligand , which forms a covalent bond with Cys721 located in the ATP-binding site of Her3. TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signalingIn VitroTX1-85-1 possesses an anti-proliferation EC 50 s of 9.9, 11.5, and 16.9 μM for Ovcar8, HCC827 GR6, and PC9 GR4 cells, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:ErbB3 23 nM (IC 50 ).

Specifications and Purity: ≥98%

Molecular Formula: C32H36N8O3

Molecular Weight: 580.7

PubChem CID: 78243752

Isomeric SMILES: CC(=O)N1CCN(CC1)C2CCC(CC2)N3C4=NC=NC(=C4C(=N3)C5=CC(=C(C=C5)OC6=CC=CC=C6)NC(=O)C=C)N

UPC:: 41116301
Condition:: New
HazmatClass:: No
WeightUOM:: LB
MPN:: T646130-1mg
CAS:: 1603845-32-4
Product Size:: 1mg

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