Biochem/physiol Actions
Specific inhibitor of MDR-1 (P-gp)
Tariquidar is a non-competitive inhibitor. It is used as a potential agent for checking the role of P-glycoprotein inhibition in cancer. Tariquidar also has an ability to enhance drug exposure in drug-resistant cancers.
Tariquidar is a potent MDR1 (P-gp, P-glycoprotein) inhibitor. Tariquidar reverses multidrug resistance (MDR) by inhibiting MDR1-mediated drug efflux.
- UPC:
- 85121805
- Condition:
- New
- HazmatClass:
- No
- MPN:
- SML1790-5MG
- CAS:
- 206873-63-4
akash.verma@cenmed.com
(732) 447-1115





