Beta gamma counters

E4031.

InformationBI-1347 BI-1347 is small molecule inhibitor of Cyclin-dependent kinase 8(CDK8) with IC50 of 1.1 nM.TargetsCDK8 (Cell-free assay) 1.1 nM.

Potent and selective BRPF1 inhibitor.

InformationGSK1838705A GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR and ALK with IC50 of 1.6 nM and 0.5 nM, respectively, and little activity to other protein kinases.In vitroGSK1838705A potently and

Glucocorticoid receptor agonist.

Glucocorticoid receptor agonist.

Potent and selective BRPF1 inhibitor.

Potent and selective BRPF1 inhibitor.

Potent and selective BRPF1 inhibitor.

Potent and selective BRPF1 inhibitor.

E4031.

E4031.