A GRP/bombesin receptor 2 antagonist (IC<sub>50</sub> = 4.13 nM in vitro) reduces bombesin-stimulated pancreatic amylase secretion and attenuates bombesin-stimulated increases in blood pressure in rats.
A GRP/bombesin receptor 2 antagonist (IC<sub>50</sub> = 4.13 nM in vitro) reduces bombesin-stimulated pancreatic amylase secretion and attenuates bombesin-stimulated increases in blood pressure in rats.
A broad-spectrum inhibitor of TACE, other ADAMs, and other MMPs inhibits PMA-induced shedding of various cell surface proteins, such as TGF-&alpha, &betaAPP, L-selectin, IL-6 receptor &alpha subunit (IC<sub>50</sub> = 10 µM) prevents
A broad-spectrum inhibitor of TACE, other ADAMs, and other MMPs inhibits PMA-induced shedding of various cell surface proteins, such as TGF-&alpha, &betaAPP, L-selectin, IL-6 receptor &alpha subunit (IC<sub>50</sub> = 10 µM) prevents
A natural anthocyanin that has neuroprotective effects, reducing amyloid &beta-induced cytotoxicity in Neuro-2A cells stimulates autophagy in U2OS cells.
A natural anthocyanin that has neuroprotective effects, reducing amyloid &beta-induced cytotoxicity in Neuro-2A cells stimulates autophagy in U2OS cells.
A potent, selective antagonist of &sigma1 receptors (Ki = 17 nM) that weakly binds &sigma2 receptors (Ki = 9,300 nM) dose-dependently inhibits neuropathic pain in several animal models, including formalin-induced nociception and capsaicin-induced
A potent, selective antagonist of &sigma1 receptors (Ki = 17 nM) that weakly binds &sigma2 receptors (Ki = 9,300 nM) dose-dependently inhibits neuropathic pain in several animal models, including formalin-induced nociception and capsaicin-induced
AD140 is an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that binds to the androgen receptor with a Ki value of 7 nM. At 0.
AD140 is an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that binds to the androgen receptor with a Ki value of 7 nM. At 0.
A selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC<sub>50</sub> values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources) potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.
A selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC<sub>50</sub> values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources) potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.
Thermal Transfer Labels for Storage in Temperatures from -40°C to 150°C For Use with Thermal Transfer Printers Unique solvent-resistant, acrylic-based adhesive provides excellent cold temperature performance Specially coated for use with a re
Thermal Transfer Labels for Storage in Temperatures from -40°C to 150°C For Use with Thermal Transfer Printers Unique solvent-resistant, acrylic-based adhesive provides excellent cold temperature performance Specially coated for use with a re
Carry out quicker start-up times Reduce your operating costs with longer lifetime amp hours Continuous light intensity for longer periods of time Data-coded and uncoded versions are available Kinesis single-element hollow cathode lamps are quick to
Carry out quicker start-up times Reduce your operating costs with longer lifetime amp hours Continuous light intensity for longer periods of time Data-coded and uncoded versions are available Kinesis single-element hollow cathode lamps are quick to