Difenidol or diphenidol

A non-selective mACh receptor antagonist and non-specific inhibitor of voltage-gated ion channels in neurons used to study animal models of vertigo and emesis.

A selective, reversible inhibitor of MAO-B (Ki = 0.091 &muM) over MAO-A (Ki = 9.06 &muM) may ameliorate depression, Parkinson&rsquos disease, Alzheimer&rsquos disease, Huntington&rsquos disease, and stroke.

A competitive antagonist of muscarinic receptors that potently blocks signaling through M1, M2, and M3 (Kis = 25, 125, and 10 nM, respectively), resulting in muscle relaxation.

A major metabolite of florfenicol, an antibiotic commonly used in veterinary medicine.

An anti-epileptic drug that inhibits the synaptosomal uptake of GABA, increasing the activation of GABAA receptors inhibits CYP3A4, CYP1A2, and CYP2C19 inhibits LDH, blocking both lactate-to-pyruvate and pyruvate-to-lactate conversions by human

A potassium channel activator that causes local relaxation in smooth muscle by increasing membrane permeability to potassium ions relaxes rat aorta rings (ED₅₀ = 19.3 &muM) and has been used as a vasodilator in the treatment of

A selective, reversible inhibitor of MAO-B (Ki = 0.091 &muM) over MAO-A (Ki = 9.06 &muM) may ameliorate depression, Parkinson&rsquos disease, Alzheimer&rsquos disease, Huntington&rsquos disease, and stroke.

A benzoylguanidine compound that selectively inhibits NHE-1 (IC₅₀s range from 0.03-3.4 &microM).

A competitive antagonist of muscarinic receptors that potently blocks signaling through M1, M2, and M3 (Kis = 25, 125, and 10 nM, respectively), resulting in muscle relaxation.

A glutamine analog that inhibits glutaminases (Ki = 6 &microM) and other glutamine-utilizing enzymes, including cytidine triphosphate synthase.

An inhibitor of SAH hydrolase (Ki = 3.9 &muM) has anti-inflammatory, anti-viral, and anti-bacterial activities.

A selective L-type calcium channel blocker with long-acting antihypertensive activity relaxes depolarization-induced contractions of rabbit aorta (EC₅₀ = 1.4 nM) and reduces the rate of spontaneously beating guinea pig right atria